122081-15-6Relevant articles and documents
TRICYCLIC GYRASE INHIBITORS
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Paragraph 0137, (2015/03/28)
Disclosed herein are compounds having the structure of Formula I and pharmaceutically suitable salts, esters, and prodrugs thereof that are useful as antibacterially effective tricyclic gyrase inhibitors. Related pharmaceutical compositions, uses and methods of making the compounds are also contemplated.
Intramolecular [2 + 2] cycloadditions of keteniminium salts derived from α- and β-amino acids. A route to azabicyclic ketones
Gobeaux, Benoit,Ghosez, Leon
, p. 29 - 32 (2007/10/02)
Unsaturated N-tosylaminoketeniminium salts generated in situ from α- and β-aminoamides readily underwent intramolecular [2 + 2]cycloadditions to give azabicyclic ketones in good yields.