155106-15-3Relevant articles and documents
Scalable and Straightforward Synthesis of All Isomeric (Cyclo)alkylpiperidines
Subota, Andrii I.,Lutsenko, Anton O.,Vashchenko, Bohdan V.,Volochnyuk, Dmitriy M.,Levchenko, Vitalina,Dmytriv, Yurii V.,Rusanov, Eduard B.,Gorlova, Alina O.,Ryabukhin, Sergey V.,Grygorenko, Oleksandr O.
, p. 3636 - 3648 (2019)
An efficient approach towards introducing (cyclo)alkyl substituents at C-2, C-3 or C-4 positions of the piperidine ring was described. The method relied on the straightforward two-step reaction sequence based on the formal sp3–sp3 re
Diastereoselective synthesis of 2-vinylpyrrolidines and 2-vinylpiperidines by the palladium-catalysed cyclization of amino-allylic carbonates containing a chiral protecting group
Olszewska, Beata,Jablonska, Aleksandra,Zawisza, Anna
, p. 254 - 271 (2018/09/10)
An efficient diastereoselective synthesis of pyrrolidine-and piperidine-type N-heterocycles is reported, by the intramolecular Pd(0)-catalysed cyclization of amino carbonates containing chiral protecting group. The use of chiral auxiliary in the cyclization gave the corresponding heterocyclic derivatives in excellent yields and with good dr values.
