194726-46-0

Basic information

• Product Name: (R)-1-(TERT-BUTOXYCARBONYL)-3-PIPERIDINECARBOXALDEHYDE
• Synonyms: (R)-1-(TERT-BUTOXYCARBONYL)-3-PIPERIDINECARBOXALDEHYDE;(R)-tert-butyl 3-formylpiperidine-1-carboxylate;tert-butyl (3R)-3-forMylpiperidine-1-carboxylate;ert-Butyl (3R)-3-formylpiperidine-1-carboxylate;tert-Butyl (R)-3-formylpiperidine-1-carboxylate;(R)-1-Boc-3-piperidinecarboxaldehyde;(R)-1-Boc-3-formyl-piperidine
• CAS NO: 194726-46-0
• Molecular Formula: C₁₁H₁₉NO₃
• Molecular Weight: 213.28
• Mol File: 194726-46-0.mol

Chemical Properties

• Appearance: /
• Density: 1.114
• Storage Temp.: Inert atmosphere,Store in freezer, under -20°C
• CAS DataBase Reference: (R)-1-(TERT-BUTOXYCARBONYL)-3-PIPERIDINECARBOXALDEHYDE(CAS DataBase Reference)
• NIST Chemistry Reference: (R)-1-(TERT-BUTOXYCARBONYL)-3-PIPERIDINECARBOXALDEHYDE(194726-46-0)
• EPA Substance Registry System: (R)-1-(TERT-BUTOXYCARBONYL)-3-PIPERIDINECARBOXALDEHYDE(194726-46-0)

Safety Data

• Hazardous Substances Data: 194726-46-0(Hazardous Substances Data)

Usage

Uses

Used in Pharmaceutical Research:
(R)-1-(TERT-BUTOXYCARBONYL)-3-PIPERIDINECARBOXALDEHYDE is used as a key intermediate in the synthesis of various pharmaceuticals and bioactive molecules. Its importance as a building block in medicinal chemistry is attributed to its ability to facilitate the creation of a wide range of functionalized piperidine derivatives for diverse biological and pharmaceutical applications.
Used in Organic Synthesis:
In the field of organic synthesis, (R)-1-(TERT-BUTOXYCARBONYL)-3-PIPERIDINECARBOXALDEHYDE serves as a versatile starting material. Its unique structure and the Boc protecting group enable the preparation of a broad spectrum of functionalized piperidine derivatives, which are essential for various applications in the chemical and pharmaceutical industries.
Used in Peptide Synthesis:
(R)-1-(TERT-BUTOXYCARBONYL)-3-PIPERIDINECARBOXALDEHYDE is utilized as a protecting agent for amine groups in peptide synthesis. The Boc group provides a stable and easily removable protection, ensuring the successful synthesis of complex peptide structures without unwanted side reactions or degradation.

Upstream product

• 116574-71-1 tert-butyl (3R)-3-(hydroxymethyl)piperidine-1-carboxylate 
• 445398-78-7 N-benzyl-hepta-4(E),6-dien-1-amine 
• 651321-53-8 Benzyl-[(E)-hepta-4,6-dien-(E)-ylidene]-amine 
• 79280-39-0 (4E)-hepta-4,6-dienal 
• 33741-15-0 methyl (4E)-hepta-4,6-dienoate 
• 934423-10-6 1-(tert-butyl)-3-methyl-(R)-piperidine-1,3-dicarboxylate 
• 24424-99-5 di-tert-butyl dicarbonate 
• 194726-40-4 (3R)-piperidine-1,3-dicarboxylic acid 1-tert-butyl ester 3-ethyl ester 

Downstream Products

• 254905-64-1 (3S)-3-(dimethylaminomethyl)piperidine-1-carboxylic acid tert-butyl ester 
• 894801-73-1 benzyl 4-{[(3S)-1-(tert-butoxycarbonyl)piperidin-3-yl]methyl}piperazine-1-carboxylate 
• 894802-13-2 tert-butyl (3S)-3-[(4-{[(3,4-dichlorophenyl)amino]carbonyl}piperazin-1-yl)methyl]piperidine-1-carboxylate 
• 116574-71-1 tert-butyl (3R)-3-(hydroxymethyl)piperidine-1-carboxylate 
• 1381949-95-6 C₂₃H₃₆N₄O₄ 
• 1381949-83-2 C₂₁H₂₉N₅O 
• 1381949-82-1 C₂₁H₂₉N₅O 
• 1381949-81-0 C₂₁H₃₂N₄O₂ 
• 894799-72-5 C₂₀H₂₉ClN₄O 
• 894799-08-7 N-(3,4-dichlorophenyl)-4-[(3R)-piperidin-3-ylmethyl]piperazine-1-carboxamide 

Relevant articles and documents

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