Journal of the American Chemical Society p. 3068 - 3073 (1998)
Update date:2022-08-04
Topics:
Aoki, Kazumasa
Peat, Andrew J.
Buchwald, Stephen L.
A new approach for the construction of indoles employing the air- and moisture-stable reagent Cp2TiCl2 is described. The key steps involved are (1) the intermolecular insertion reactions of an olefin and a titanocene- stabilized benzyne complex and (2) the Pd-catalyzed aryl amination reaction. The simplicity and availability of the requisite starting materials give the method a broad scope for the preparation of polysubstituted indoles.
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