Chinese Chemical Letters p. 253 - 256 (2010)
Update date:2022-08-03
Topics:
Tang, Peng Cho
Lin, Zhi Gang
Wang, Yang
Yang, Fang Long
Wang, Qian
Fu, Jian Hong
Zhang, Lei
Gong, Ai Shen
Luo, Jing Jing
Dai, Jun
She, Gao Hong
Si, Dan Dan
Feng, Jun
An efficient stereoselective synthesis of the rigid aza-bicyclo[3.2.0]heptane scaffold has been developed to provide 2-cyano pyrrolidine alpha-amino amide 1 as DPP-4 inhibitor.
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