ENANTIOSELECTIVE TOTAL SYNTHESIS OF GLYOXALASE I INHIBITOR USING ASYMMETRIC DIELS-ALDER REACTION OF A NEW CHIRAL DIENOPHILE, (S)S-3-(3-TRIFLUOROMETHYLPYRID-2-YLSULFINYL)ACRYLATE.

DOI: 10.1016/S0040-4039(00)85252-1

Source and publish data:

Tetrahedron Letters p. 5509 - 5512 (1986)

Update date:2022-07-29

Topics:

Authors:

Takayama, Hiromitsu

Hayashi, Kazuya

Koizumi, Toru

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Article abstract of DOI:10.1016/S0040-4039(00)85252-1

Highly enantioselective total synthesis of Glyoxalase I inhibitor (1) was achieved utilizing the assymetric Diels-Alder reaction of a new chiral dienophile, (S)_S-menthyl 3-(3-trifluoromethylpyrid-2-ylsulfinyl)acrylate (3) with 2-methoxyfuran.

Full text of DOI:10.1016/S0040-4039(00)85252-1

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