
Journal of Medicinal Chemistry p. 798 - 806 (2009)
Update date:2022-08-04
Topics:
Sugimoto, Yoshinori
Konoki, Keiichi
Murata, Michio
Matsushita, Masafumi
Kanazawa, Hiroshi
Oishi, Tohru
Salicylihalamide A (SA), a benzolactone enamide compound, possesses potent cytotoxicity against human tumor cell lines. SA is a selective inhibitor of mammalian vacuolar type H+-ATPase (V-ATPase), and is distinct from previously known V-ATPase
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