Journal of Medicinal Chemistry p. 176 - 181 (1988)
Update date:2022-08-04
Topics:
Bock, Mark G.
DiPardo, Robert M.
Evans, Ben E.
Rittle, Kenneth E.
Veber, Daniel F.
et al.
A series of 4-substituted 4H-<1,2,4>triazolo<4,3-a><1,4>benzodiazepines was prepared by standard metodology.These compounds were tested in vitro as antagonists of the binding of <125I>cholestokinin (CCK) to rat pancreas and guinea pig brain receptors and
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