Analogues of oxytocin with an oxime bridge using chemoselectively addressable building blocks

Article abstract of DOI:10.1016/0040-4039(96)01537-7

The synthesis of two novel amino-acid building blocks for the chemoselective ligation of unprotected peptides via oxime bond formation and their application in the solid phase peptide synthesis of oxytocin analogues with the disulfide altered to an oxime bridge are described.