Selective [3 + 2] huisgen cycloaddition. Synthesis of TVaws-disubstituted triazolodiazepines from asa-baylis-hillman adducts

DOI: 10.1021/jo802533d

Source and publish data:

Journal of Organic Chemistry p. 2004 - 2007 (2009)

Update date:2022-08-05

Topics:

Authors:

Declerck, Valerie

Toupet, Loic

Martinez, Jean

Lamaty, Frederic

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jo802533d

The 1,3-dipolar cycloaddition of linear azido alkynes derived from protected β-amino esters proceeds via diastereomeric differentiation to provide irans-disubstituted triazolodiazepines in good yields.

Full text of DOI:10.1021/jo802533d

Products guided by the article

Product name:C₁₉H₂₇NO₄SSi

Cas No:1123303-63-8

R&D Labs maybe for 1123303-63-8

Kaiping Genuine Biochemical Pharmaceutical Co.,Ltd.

Contact:+86-750-2881198

Address:No.1, Xinke Road, Shatang Town, Kaiping, Guangdong Province, P.R.China
Shanghai Norky Pharmaceutical Co., LTD.

website:http://www.norkypharm.com

Contact:86-21-61075300

Address:1165 Jiangning Road, Office 1502, Shanghai, China
NINGBO PANGS CHEM INT’L CO., LTD.

Contact:+86-0574-27666801

Address:Floor 21, Building 11, Xintiandi, No. 689, Shijiroad, Ningbo, Zhejiang, China
Nanjing Chemical Material Corp.(NCMC)

website:http://www.njchemm.com

Contact:0086-25-83172879

Address:B12 Technology and Innovation Building, Nanjing Tech University, No.5 New Model Road
Oren Hydrocarbons (Qingdao) Co., Ltd.

Contact:+86-532-68607667-801

Address:Room 3 # 302, No.9 Qingyun Road, Qingdao, China

Relevant to this article

Regioselective Chlorination and Suzuki–Miyaura Cross-Coupling of 4-Alkoxycoumarins, 4-Alkoxy-2-pyrones, and Related Heterocycles

Doi:10.1002/ejoc.201700837
(2017)
Synthetic and theoretical investigations on the construction of oxanorbornenes by a Michael addition and intramolecular Diels-Alder furan reaction

Doi:10.1002/ejoc.200800681
(2008)
ANTIINFLAMMATORY ACTIVITY OF 3,4-DISUBSTITUTED PYRAZOLES

Doi:10.1007/BF00758133
(1987)
Diastereoselective synthesis of polycyclic acetal-fused pyrano[3,2-c]pyran-5(2H)-one derivatives

Doi:10.1021/jo8023889
(2009)
STEREOCHEMISCHE ASPEKTE IN ZUSAMMENHANG MIT DER SYNTHESE VON 2,6-ANHYDRO-1-DESOXY-1-NITROALDITOLEN

Doi:10.1016/0008-6215(87)80143-X
(1987)
Synthesis of building blocks for the development of the SUPRAPhos ligand library and examples of their application in catalysis

Doi:10.1002/ejoc.200800499
(2008)

Article Doi