N-[(Dihydroxyphenyl)acyl]serotonins as potent inhibitors of tyrosinase from mouse and human melanoma cells

DOI: 10.1016/j.bmcl.2009.05.115

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 4178 - 4182 (2009)

Update date:2022-08-05

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Authors:

Yamazaki, Yoshimitsu

Kawano, Yasuhiro

Yamanaka, Akiko

Maruyama, Susumu

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Article abstract of DOI:10.1016/j.bmcl.2009.05.115

A series of N-acyl derivatives of tyramine, tryptamine, and serotonin were synthesized and tested on anti-melanogenic activity. The serotonin derivatives such as N-caffeoylserotonin (3) and N-protocatechuoylserotonin (9) were inhibitory to tyrosinase from

Full text of DOI:10.1016/j.bmcl.2009.05.115

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