Stereospecific synthesis of a-substituted syn-α,β-diamino acids by the diaza-cope rearrangement

DOI: 10.1021/ol9021904

Source and publish data:

Organic Letters p. 5258 - 5260 (2009)

Update date:2022-08-05

Topics:

Authors:

Kim, Hyunwoo

Chin, Jik

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Article abstract of DOI:10.1021/ol9021904

Diaza-Cope rearrangement is used to make a variety of a-substituted syn-α,β-diamino acids. The rearrangement takes place with complete transfer of stereochemical integrity (>97% de and >98% ee) giving only one of four possible stereoisomers as determined

Full text of DOI:10.1021/ol9021904

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