One-pot synthesis of unsymmetrical 2,3-diarylindoles by site-selective suzuki-miyaura reactions of N -methyl-2,3-dibromoindole

Article abstract of DOI:10.1055/s-0029-1219201

The Suzuki-Miyaura reaction of N-methyl-2,3-dibromoindole with two equivalents of boronic acids gave symmetrical 2,3-diarylindoles. The reaction with one equivalent of arylboronic acid resulted in site-selective formation of 2-aryl-3-bromoindoles. The one