Synthesis and biological evaluation of 14-alkoxymorphinans. 3. Extensive study on cyprodime-related compounds

DOI: 10.1021/jm00166a018

Source and publish data:

Journal of Medicinal Chemistry p. 1200 - 1206 (1990)

Update date:2022-08-03

Topics:

Authors:

Schmidhammer

Smith Smith

Erlach Erlach

Koch Koch

Krassnig

Schwetz Schwetz

Wechner Wechner

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Article abstract of DOI:10.1021/jm00166a018

A series of cyprodime-related compounds (2, 4-12, and 26) has been synthesized and evaluated for opioid agonist and antagonist activity with the mouse vas deferens and guinea pig ileum preparations. None of the changes to cyprodime, including the introduc

Full text of DOI:10.1021/jm00166a018

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