Bioorganic and Medicinal Chemistry Letters p. 6286 - 6290 (2010)
Update date:2022-08-04
Topics:
Corminboeuf, Olivier
Bezenon, Olivier
Grisostomi, Corinna
Remeň, ?ubo?
Richard-Bildstein, Sylvia
Bur, Daniel
Prade, Lars
Hess, Patrick
Strickner, Panja
Fischli, Walter
Steiner, Beat
Treiber, Alexander
The discovery of a new series of piperidine-based renin inhibitors is described herein. SAR optimization upon the P3 renin sub-pocket is described, leading to the discovery of 9 and 41, two bioavailable renin inhibitors orally active at low doses in a tra
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