1-(Aminoalkyl)-2-phenylindoles as novel pure estrogen antagonists

DOI: 10.1021/jm00171a045

Source and publish data:

Journal of Medicinal Chemistry p. 2635 - 2640 (1990)

Update date:2022-07-30

Topics:

Authors:

Von Angerer

Knebel Knebel

Kager Kager

Ganss Ganss

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Article abstract of DOI:10.1021/jm00171a045

A number of 1-(ω-aminoalkyl)-5-hydroxy-2-(4-hydroxyphenyl)indoles were synthesized and studied for their binding affinities for the calf uterine estrogen receptor and estrogen antagonistic activities. Highest binding affinities were found with derivatives

Full text of DOI:10.1021/jm00171a045

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