Studies on Neurokinin Antagonists. 2. Design and Structure-Activity Relationships of Novel Tripeptide Substance P Antagonists, Nα-α-(Nα-Acetyl-L-threonyl)-N1-formyl-D-tryptophyl>-N-methyl-N-(phenylmethyl)-L-ph

DOI: 10.1021/jm00095a013

Source and publish data:

Journal of Medicinal Chemistry p. 3184 - 3191 (1992)

Update date:2022-08-05

Topics: Substance P Methyl Tripeptide N-terminal

Authors:

Hagiwara, Daijiro

Miyake, Hiroshi

Morimoto, Hiroshi

Murai, Masako

Fujii, Takashi

Matsuo, Masaaki

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Article abstract of DOI:10.1021/jm00095a013

Continuing studies on the chemical modification of the previously reported novel tripeptide SP antagonist, N^α-α-α-(tert-butyloxycarbonyl)glutaminyl>-N¹-formyl-D-tryptophyl>phenylalanine benzyl ester View More

Full text of DOI:10.1021/jm00095a013

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