Studies on antiulcer drugs. III. Synthesis and antiulcer activities of imidazo[1,2-a]pyridinylethylbenzoxazoles and related compounds. A novel class of histamine H2-receptor antagonists.

DOI: 10.1248/cpb.40.1424

Source and publish data:

Chemical and pharmaceutical bulletin p. 1424 - 1438 (1992)

Update date:2022-08-03

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Authors:

Katsura Katsura

Inoue Inoue

Nishino Nishino

Tomoi Tomoi

Itoh Itoh

Takasugi

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Article abstract of DOI:10.1248/cpb.40.1424

A series of imidazo[1,2-a]pyridinylalkylbenzoxazole derivatives was synthesized and tested for histamine H2-receptor antagonist, gastric antisecretory and antiulcer activities. Some of 2-amino-6-[2-(imidazo[1,2-a]pyridin-2-yl)ethyl]benzoxazole derivatives

Full text of DOI:10.1248/cpb.40.1424

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