Thiophene systems. 12. Analogues of ketanserin and ritanserin as selective 5-HT2 antagonists

DOI: 10.1016/0223-5234(91)90007-A

Source and publish data:

European Journal of Medicinal Chemistry p. 807 - 813 (1991)

Update date:2022-08-03

Topics: Thiophene Antagonists Analogues

Authors:

Press, JB

Russell, RK

McNally, JJ

Rampulla, RA

Falotico, R

et al. et al.

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Article abstract of DOI:10.1016/0223-5234(91)90007-A

A series of thieno<3,2-d>-, <4,3-d>- and <2,3-d>pyrimidinedione derivatives was prepared with N-3 substitution containing the side chains of ketanserin and ritanserin.The best of these thiophene analogues were the isosteres of ketanserin which were up to

Full text of DOI:10.1016/0223-5234(91)90007-A

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