Thiophene systems. 12. Analogues of ketanserin and ritanserin as selective 5-HT2 antagonists

DOI: 10.1016/0223-5234(91)90007-A

Source and publish data:

European Journal of Medicinal Chemistry p. 807 - 813 (1991)

Update date:2022-08-03

Topics: Thiophene Antagonists Analogues

Authors:

Press, JB

Russell, RK

McNally, JJ

Rampulla, RA

Falotico, R

et al. et al.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0223-5234(91)90007-A

A series of thieno<3,2-d>-, <4,3-d>- and <2,3-d>pyrimidinedione derivatives was prepared with N-3 substitution containing the side chains of ketanserin and ritanserin.The best of these thiophene analogues were the isosteres of ketanserin which were up to

Full text of DOI:10.1016/0223-5234(91)90007-A

Products guided by the article

Product name:Thieno[3,4-d]pyrimidine-2,4(1H,3H)-dione, 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-

Cas No:130501-99-4

R&D Labs maybe for 130501-99-4

Shanghai Hohance Chemical Co., ltd

Contact:13914753421

Address:Fl.5；Bld. 70, Lane 1500; Xinfei Road
Beijing Stable Chemcial Co.ltd

Contact:86-10-63785052

Address:A1301 Technological Edifice. No.4 FuFeng Road,FengTai District, Beijing. China
Jining Shengrun Chemical Industry Co., Ltd.

Contact:+86-537-7121666 ,

Address:West Ring Road,Wenshang County Shandong Province
Taizhou Green Peptide Trading Co., Ltd.

Contact:--

Address:Room 1501, No71, Yuehe Road, Taizhou City, Zhejiang Province, China
HAORUI ENTERPRISES LLC

Contact:(1) 206-3550089

Address:5115 NE 8TH PL, Renton, WA 98059 USA

Relevant to this article

Unusual reactivity of azomethine ylides due to electronic effects: A novel route to 5-alkylidene-3-oxazolines

Doi:10.1016/S0040-4039(00)89060-7
(1990)
Stereoselective synthesis of trans-1,2-di-O-acetyl glycoses

Doi:10.1055/s-1990-26995
(1990)
Low-Valent Titanium Induced Reductive Cyclization of Nitriles to Symmetrically Substituted Tetraalkylpyrazines

Doi:10.1055/s-1990-26987
(1990)
The novel triazine cored tripodal and trinuclear Schiff base-oxime metal complexes: Their magnetic properties and thermal decompositions

Doi:10.1002/jhet.671
(2011)
Practical and highly stereoselective method for the preparation of several chiral arylsulfinamides and arylsulfinates based on the spontaneous crystallization of diastereomerically pure N-benzyl-N-(1-phenylethyl)- arylsulfinamides

Doi:10.1016/j.tetasy.2011.01.028
(2011)
Microwave-assisted aliphatic fluorine-chlorine exchange using triethylamine trihydrofluoride (TREAT-HF)

Doi:10.1016/j.tetlet.2009.03.103
(2009)

Article Doi