THE SYNTHESIS OF (+)- AND (-)-1-BENZOYL-1,2,2a,3,4,5-HEXAHYDROBENZINDOL-4-AMINE, and PREPARATION OF LY228729

DOI: 10.1016/S0040-4039(00)97303-9

Source and publish data:

Tetrahedron Letters p. 7579 - 7582 (1990)

Update date:2022-07-29

Topics:

Authors:

Martinelli, Michael J.

Leanna, M. Robert

Varie, David L.

Peterson, Barry C.

Kress, Thomas J.

et al. et al.

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Article abstract of DOI:10.1016/S0040-4039(00)97303-9

Racemic epoxide 5 was reacted with S-Phenylethylamine to afford diastereomers 6 and 7, from which amino alcohol 6 could be isolated directly.Aziridine formation and tandem-hydrogenolysis provided optically pure primary amine 2 (31percent from racemic 4),

Full text of DOI:10.1016/S0040-4039(00)97303-9

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