A NOVEL SUBSTITUTION REACTION OF 4-SULFINYLAZETIDIN-2-ONE WITH SILYLATED HETERONUCLEOPHILES: AN EFFICIENT SYNTHESIS OF 4-HETEROFUNCTION SUBSTITUTED 3-(1-HYDROXY)ETHYLAZETIDIN-2-ONES

DOI: 10.1016/S0040-4039(00)79927-8

Source and publish data:

Tetrahedron Letters p. 2375 - 2378 (1991)

Update date:2022-08-02

Topics:

Authors:

Kita, Yasuyuki

Shibata, Norio

Yoshida, Naoki

Tohjo, Takashi

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)79927-8

4-Sulfinylazetidin-2-one was reacted with silylated heteronucleophiles in the presence of a catalytic amount of zinc iodide to give the corresponding trans-4-heterofunction substituted azetidin-2-ones in high yields.

Full text of DOI:10.1016/S0040-4039(00)79927-8

Products guided by the article

Product name:(3R,4R)-3-<(1R)-(1-tert-butyldimethylsiloxy)ethyl>-4-(2-phenylbutyroyloxy)azetidin-2-one

Cas No:134987-72-7

R&D Labs maybe for 134987-72-7

Weifang Adde Economic And Trade Co.,LTD.

Contact:86-536-8885548

Address:Room 1402,Wanda Plaza B Block,No.958,Yuanfei Road,Kuiwen District
Arshine Pharmaceutical Co., Limited

website:http://www.cnarshine.com

Contact:0731-88503671

Address:Room 1109.Block C3, Lugu Enterprise Plaza,No.27 Wenxuan Road,Changsha National Hi-Tech Industrial Development Zone,Hunan ,P.R.China
Wuhan Shangrisyn chemicals Technology Co.,Ltd(expird)

Contact:+86-027-84466317 __ +86-15387123698

Address:wuhan - china
Suns Chemical Sdn Bhd

Contact:0086 371 65711996

Address:Jalan 4/3, Kawasan Perindustrian Serendah, 48000 Rawang,
ORCHID CHEMICAL SUPPLIES LTD

website:http://www.orchid-chem.com

Contact:+86-571-85395792

Address:607, North Zhongshan Road, Hangzhou 310000 China

Relevant to this article

Total syntheses of ent-heliespirones A and C

Doi:10.1021/jo201971g
(2012)
Synthesis of mixed N,N′-(Ar,Ar′-diaryl)iminoisoindolines for applications in palladacycle formations

Doi:10.1016/j.ica.2011.09.054
(2011)
One-pot synthesis of functionalized α-acyloxythioamides from N-protected a-amino acids as an acid component in the Passerini reaction in an ionic liquid

Doi:10.1007/BF03245894
(2011)
Convenient synthesis of α-terthienyl and α-quinquethienyl via a Friedel-Crafts route

Doi:10.1055/s-1991-26494
(1991)
Hydrophosphonylation of alkenes or nitriles by double radical transfer mediated by titanocene/propylene oxide

Doi:10.1016/j.tetlet.2011.09.096
(2011)
Inhibitors of HIV-1 maturation: Development of structure-activity relationship for C-28 amides based on C-3 benzoic acid-modified triterpenoids

Doi:10.1016/j.bmcl.2016.03.019
(2016)

Article Doi