Tetrahedron Letters p. 5831 - 5834 (1993)
Update date:2022-07-30
Topics:
Desai, Manoj C.
Thadeio, Peter F.
Lefkowitz, Sheri L.
The synthesis of racemic CP-99,994, a highly potent substance P antagonist is reported. The synthesis outlined here is suitable for developing structure activity relationships for this important class of compounds.
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