Synthesis of (±)-CP-99994: A highly potent substance P antagonist

DOI: 10.1016/S0040-4039(00)73791-9

Source and publish data:

Tetrahedron Letters p. 5831 - 5834 (1993)

Update date:2022-07-30

Topics:

Authors:

Desai, Manoj C.

Thadeio, Peter F.

Lefkowitz, Sheri L.

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Article abstract of DOI:10.1016/S0040-4039(00)73791-9

The synthesis of racemic CP-99,994, a highly potent substance P antagonist is reported. The synthesis outlined here is suitable for developing structure activity relationships for this important class of compounds.

Full text of DOI:10.1016/S0040-4039(00)73791-9

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