Synthesis, pharmacological investigation and computational studies on a tricyclic ergoline analog with selective dopamine autoreceptor activity

DOI: 10.1002/ardp.19953280708

Source and publish data:

Archiv der Pharmazie p. 609 - 614 (1995)

Update date:2022-09-26

Topics:

Authors:

Gmeiner Gmeiner

Bollinger

Mierau Mierau

Hofner Hofner

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Article abstract of DOI:10.1002/ardp.19953280708

The novel aminobenzindolone 8 was prepared and evaluated as a potential antipsychotic agent. The target compound was synthesized in eight steps starting from the tetrahydrobenzindolone 9. The key step of the synthesis was an electrophilic amination of the

Full text of DOI:10.1002/ardp.19953280708

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