Ring transformation with bridged 1,3-dicarbonyl heteroanalogues, III. 5-(ω-aminoalkyl)-1,2,4-oxadiazoles by ring-transformations of 3-methylthio-2-aza-3-propeniminium salts

DOI: 10.1002/ardp.2503241205

Source and publish data:

Archiv der Pharmazie p. 963 - 965 (1991)

Update date:2022-08-04

Topics: Experimental terms Ring transformation

Authors:

Patzel Patzel

Liebscher

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1002/ardp.2503241205

3-Methylthio-2-aza-3-propeniminium salts 5 react with hydroxylamine after ring transformation under formation of 5-(ω-aminoalkyl)-1,2,4-oxadiazole hydroiodides 4·HI, which show a remarkable antitussive activity.

Full text of DOI:10.1002/ardp.2503241205

Products guided by the article

Product name:[5-(3-Methylamino-propyl)-[1,2,4]oxadiazol-3-yl]-phenyl-amine; hydriodide

Cas No:138970-13-5

R&D Labs maybe for 138970-13-5

HANGZHOU TOYOND BIOTECH CO., LTD

Contact:+86-571-86965177

Address:No. 189, Fengqi East Road, Hangzhou, China
Huayi Isotopes Co.

Contact:+ 86 512 52491118

Address:1 Fuyu Road, Haiyu TownChangshu, Jiangsu, China
Anhui Gusheng Import&Export CO.,LTD

Contact:86-551-63662296

Address:Jinzhai Road NO.162 ,hefei, china
Rely Chemicals Ltd.

Contact:+86-518-81061113

Address:No. 8 Lingzhou Road, Lianyungang, Jiangsu, China
Dongguan Albiya Energy Science and Technology Co.,Ltd

Contact:+86-769-22181286

Address:Huanan Industial Park, Dongguan,China

Relevant to this article

Synthesis of 11-Amino-substituted-5,6-dimethyl-5H-pyrido<3',4':4,5>pyrrolo<2,3-g>isoquinolines as New Ellipticine Analogues

Doi:10.1039/P19910003173
(1991)
Synthesis and antinociceptive activity of [D-Ala²]Leu-enkephalin derivatives conjugated with the adamantane moiety

Doi:10.1248/cpb.45.1782
(1997)
Organocatalyzed Michael-Henry reactions: Enantioselective synthesis of cyclopentanecarbaldehydes via the dienamine organocatalysis of a succinaldehyde surrogate

Doi:10.1039/c2cc33309k
(2012)
Microwave-assisted solvent-free synthesis of 2-styrylquinolines in the presence of zinc chloride

Doi:10.1134/S1070428012060139
(2012)
Click fleximers: A modular approach to purine base-expanded ribonucleoside analogues

Doi:10.1039/c2ob25678a
(2012)
Design, synthesis and antiproliferative activity of novel 2-substituted-4-amino-6-halogenquinolines

Doi:10.3390/molecules17055870
(2012)

Article Doi