Asymmetric Aza-Diels-Alder Reaction Mediated by Chiral Boron Reagent

DOI: 10.1021/jo00038a003

Source and publish data:

Journal of Organic Chemistry p. 3264 - 3265 (1992)

Update date:2022-08-03

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Authors:

Hattori, Kouji

Yamamoto, Hisashi

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Article abstract of DOI:10.1021/jo00038a003

An asymmetric aza-Diels-Alder reaction of an imine mediated by an in situ generated chiral boron complex is described.The method is successful with several aldimines and affords products of up to 90percent ee.

Full text of DOI:10.1021/jo00038a003

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