Asymmetric Aza-Diels-Alder Reaction Mediated by Chiral Boron Reagent

DOI: 10.1021/jo00038a003

Source and publish data:

Journal of Organic Chemistry p. 3264 - 3265 (1992)

Update date:2022-08-03

Topics:

Authors:

Hattori, Kouji

Yamamoto, Hisashi

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jo00038a003

An asymmetric aza-Diels-Alder reaction of an imine mediated by an in situ generated chiral boron complex is described.The method is successful with several aldimines and affords products of up to 90percent ee.

Full text of DOI:10.1021/jo00038a003

Products guided by the article

Product name:N-benzyl-2,3-dihydro-2-(c-hexyl)-5-methyl-4-pyridone

Cas No:141120-52-7

R&D Labs maybe for 141120-52-7

Sichuan Mianzhu Ronghong Chemical Co.,LTd

Contact:8613981840544

Address:XINSHI INDUSTRY PARK,MIANZHU,SICHUAN,CHINA
Ji'nan Orgachem Pharmaceutical Co.,Ltd

Contact:+86-531-82687810

Address:Jinan
BAODING SINO-CHEM INDUSTRY CO.,LTD

Contact:0312-5956088

Address:NO.8 FUXING ROAD,CHINA
AstaTech ( Chengdu) BioPharmaceutical Corp.

website:http://www.astabiochem.cn/

Contact:+86-15198215156-15198215156

Address:SICHUAN CHENGDU
LIAONING DMSO CHEMICALS CO.,LTD.

website:http://www.chinadmso.com

Contact:+86-427-6503033

Address:FLOOR 16, BLOCK A, FINANCIAL SQUARE, XINGLONGTAI DISTRICT, PANJIN CITY, LIAONING P.R. CHINA

Relevant to this article

New reactions of quaternary ammonium salts derived from vinamidinium salt reduction products and a reassignment of structure

Doi:10.1080/00397919208019298
(1992)
Ni-Catalyzed Reductive Allylation of α-Chloroboronates to Access Homoallylic Boronates

Doi:10.1021/acs.orglett.1c01213
(2021)
Sulphonamide and sulphonyl-hydrazone cyclic imide derivatives: Antinociceptive activity, molecular modeling and in Silico ADMET screening

Doi:10.1007/s12272-012-1002-1
(2012)
Design, synthesis and pharmacological characterization of coumarin-based fluorescent analogs of excitatory amino acid transporter subtype 1 selective inhibitors, UCPH-101 and UCPH-102

Doi:10.1016/j.bmc.2012.09.049
(2012)
Synthesis, biological evaluation, and molecular modeling of donepezil and N-[(5-(Benzyloxy)-1-methyl-1H-indol-2-yl)methyl]-N-methylprop-2-yn-1-amine hybrids as new multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer's disease

Doi:10.1021/jm200853t
(2011)
Synthesis and screening of 2-(2-(4-substituted piperazine-1-yl)-5- phenylthiazol-4-yl)-3-aryl quinazolinone derivatives as anticancer agents

Doi:10.1007/s00044-012-0260-2
(2013)

Article Doi