Para-substituted Phe3 deltorphin analogues: Enhanced selectivity of halogenated derivatives for δ opioid receptor sites

DOI: 10.1021/jm00103a001

Source and publish data:

Journal of Medicinal Chemistry p. 4651 - 4657 (1992)

Update date:2022-08-04

Topics:

Authors:

Salvadori

Bianchi Bianchi

Lazarus Lazarus

Scaranari

Attila Attila

Tomatis Tomatis

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00103a001

The δ-selective opioid peptide deltorphin C(H-Tyr-D-Ala-Phe-Asp-Val-Val- Gly-NH₂) (DEL C) was modified by para-substitution of Phe³ with halogens (F, Cl, Br, I), amino, or nitro groups. The bioactive potencies in peripheral tissues a

Full text of DOI:10.1021/jm00103a001

Products guided by the article

Product name:Boc-Tyr-D-Ala-p-NO₂Phe-Glu(OtBu)-Val-Val-Gly-NH₂

Cas No:145277-73-2

R&D Labs maybe for 145277-73-2

Wuxi Innopal International Trade CO.,LTD

Contact:+86-510-80711901-8003

Address:Room 402,Building 5,Longze Garden,No.17,South huanjiu Road,Yixing City, Jiangsu,China
Shenzhen Sungening Medicine Co., Ltd

Contact:+86-871-65110906

Address:Room702, Building 2, 365 Dianchi Road, Kunming, Yunnan Province, P.R. China
Shenyang Xingzhenghe Chemical Co., Ltd.

Contact:024-23509232

Address:No. 33, Naner Road, Heping Dist.
Jiangsu Taihu New Materials Holding Co., Ltd

Contact:+86-519-86160108

Address:Xueyan Town, Changzhou City, Jiangsu Province, 213169, China
TIANJIN DONGRUXIANG MINERALS MARKETING CO.,LTD(expird)

Contact:22-58516360

Address:tianjin

Relevant to this article

Highly enantioselective intermolecular hydroamination of allylic amines with chiral aldehydes as tethering catalysts

Doi:10.1002/chem.201203462
(2013)
Biotransformation of artemisinin derivatives by Glycyrrhiza glabra, Lavandula officinalis, and Panax quinquefolium

Doi:10.1007/s00044-013-0726-x
(2014)
Iminopropadienones, RN=C=C=C=O: Syntheses and Reactions

Doi:10.1039/c39920001571
(1992)
One-pot asymmetric synthesis of 2-aryl-2,3-dihydro-4-quinolones catalyzed by amino acid-derived sulfonamides

Doi:10.1016/j.tetasy.2013.05.028
(2013)
Synthesis of novel geldanamycin derivatives

Doi:10.1016/j.tet.2021.131927
(2021)
Identification of the KDM2/7 histone lysine demethylase subfamily inhibitor and its antiproliferative activity

Doi:10.1021/jm400624b
(2013)

Article Doi