Enantioselektive Synthese von Allyl-, Propargyl- und 4-En-2-inyl-aminen durch 1,2-Addition von Organocer-Reagenzien an chirale Aldimine

DOI: 10.1002/hlca.19950780419

Source and publish data:

Helvetica Chimica Acta p. 970 - 992 (1995)

Update date:2022-08-02

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Authors:

Enders, Dieter

Schankat, Juergen

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Article abstract of DOI:10.1002/hlca.19950780419

(E)- and (Z)-Allyl-, propargyl, and 4-en-2-ynyl-amines 5 and 14, useful bifunctional building blocks and of pharmaceutical interest, are synthesized in high enantiomeric purity (e.e. >/= 97 percent).Key step is the diastereoselective 1,2-addition (d.e. 86

Full text of DOI:10.1002/hlca.19950780419

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