3-Substituted, 3-(4-pyridinylmethyl)-1,3-dihydro-1-phenyl-2H-indol-2-ones as acetylcholine release enhancers: Synthesis and SAR

DOI: 10.1021/jm00072a009

Source and publish data:

Journal of Medicinal Chemistry p. 2899 - 2907 (1993)

Update date:2022-08-05

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Authors:

Wilkerson

Kergaye Kergaye

Tam Tam

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Article abstract of DOI:10.1021/jm00072a009

A series of 3-substituted, 3-(4-pyridinylmethyl)-1,3-dihydro-1-phenyl-2H- indol-2-ones was synthesized and found to enhance the stimulus-induced release of neurotransmitter acetylcholine (AcCh), and by doing so, might be useful in treating cognitive disor

Full text of DOI:10.1021/jm00072a009

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Product name:2,3-dihydro-2-oxo-1-phenyl-3-(4-pyridinylmethyl)-1H-indole-3-butanoic acid ethyl ester

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