Journal of Medicinal Chemistry p. 1015 - 1027 (1994)
Update date:2022-08-04
Topics:
Trinks
Buchdunger
Furet
Kump
Mett
Meyer
Muller
Regenass
Rihs
Lydon
Traxler
Dianilinophthalimides represent a novel class of inhibitors of the EGF- receptor protein tyrosine kinase with a high degree of selectivity versus other tyrosine and serine/threonine kinases. Steady-state kinetic analysis of compound 3, which showed potent
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Doi:10.1016/S0040-4039(01)99639-X
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(1994)