
Synthetic Communications p. 2215 - 2221 (1994)
Update date:2022-08-05
Topics:
Ten Hoeve
Wynberg
Cyclic amidines are prepared in 3 steps from an aromatic aldehyde, isobutyraldehyde, and urea. The amidines 1 and 2 are readily resolved using chiral cyclic phosphoric acids.
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Doi:10.1039/DT9790000715
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(1994)Doi:10.1021/om5003182
(2014)Doi:10.1002/anie.201309847
(2014)