N-(4-Nitrophenyl)oxamic acid and related N-acylanilines are non-competitive inhibitors of Vibrio cholerae sialidase but do not inhibit Trypanosoma cruzi or Trypanosoma brucei trans-sialidases

DOI: 10.1002/hlca.19940770425

Source and publish data:

Helvetica Chimica Acta p. 1166 - 1174 (1994)

Update date:2022-07-30

Topics:

Authors:

Engstler

Ferrero-Garcia

Parodi Parodi

Schauer Schauer

Storz-Eckerlin

Vasella Vasella

Witzig Witzig

Zhu Zhu

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Article abstract of DOI:10.1002/hlca.19940770425

N-(4-Nitrophenyl)oxamic acid 1, N-(2-fluoro-4-nitrophenyl)oxamic acid 7, N-(4-nitrophenyl)trifluoroacetamide 3, and N-(2-methoxy-4-nitrophenyl)trifluoroacetamide 9 are non-competitive inhibitors of Vibrio cholerae sialidase with K(i)-values ranging from 2

Full text of DOI:10.1002/hlca.19940770425

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