Studies on a novel, potent and orally effective cholecystokinin A antagonist, FK-480. Synthesis and structure-activity relationships of FK-480 and related compounds

DOI: 10.1248/cpb.42.2071

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 2071 - 2083 (1994)

Update date:2022-07-30

Topics:

Authors:

Satoh Satoh

Matsuo Matsuo

Sogabe Sogabe

Itoh Itoh

Tada Tada

Kinoshita

Yoshida Yoshida

Takaya Takaya

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.42.2071

We prepared various novel tricyclic 1,4-benzodiazepine derivatives as cholecystokinin (CCK) A antagonists, which were evaluated preliminarily for inhibition of ¹²⁵I-CCK-8 binding to rat pancreatic membranes in vitro and inhibiting effect on CCK

Full text of DOI:10.1248/cpb.42.2071

NII-Electronic Library Service

Products guided by the article

Product name:(3,4-Dihydro-2H-benzo[1,4]thiazin-5-yl)-(2-fluoro-phenyl)-methanone

Cas No:163155-61-1

R&D Labs maybe for 163155-61-1

Suzhou ATL Chemical Co.,ltd

Contact:+86-0512-69209969

Address:Room 317,Lushan Road,Suzhou New District,Jiangsu Province,China.
Xinjiang Zhongtai Chemical Co., Ltd.

Contact:+86-991-8788172

Address:NO.78 XISHAN RD.URUMQI，CHINA
Brichem ( Haikou ) Co. Ltd.

Contact:86-898-65311214

Address:Room 102, BLDG. 68 Jiangnan City, No. 66 Heping Road,Haikou, Hainan, China
Jiangxi Lanqi Fine Chemical S&T Co., Ltd.

Contact:+86-21-64891143

Address:XinJiShan Industrial Area, Zhangshu City, JiangXi Province, China
Shanghai Yingrui Biopharma Co., Ltd

Contact:021-3358 8661*8003

Address:shanghai

Relevant to this article

Doi:10.1016/0008-6215(67)85013-4
(1967)
Design, synthesis, structure-activity relationship and insecticidal activities of trifluoromethyl-containing sulfiliminyl and sulfoximinyl phthalic acid diamide structure

Doi:10.1002/cjoc.201400223
(2014)
A general synthetic route to anomeric α-azido and α-amino acids and formal synthesis of (+)-hidantocidin

Doi:10.1021/jo00103a057
(1994)
Antibody-catalyzed rearrangement of a peptide bond: Mechanistic and kinetic investigations

Doi:10.1021/ja00122a001
(1995)
Polycyclic N-heterocyclic compounds 76: Synthesis and antiplatelet evaluation of 2,4-disubstituted 5,6-Dihydro[1]benzofuro[3′,2′:2,3] oxepino[4,5-d]pyrimidines

Doi:10.1002/jhet.1539
(2014)
Aromatic phosphonate-phosphines

Doi:10.1080/10426509608038791
(1996)

Hot Product

65-85-0
624-28-2
30123-17-2
108-67-8
50-28-2
71-58-9
75980-60-8
2687-91-4 N-Ethyl Pyrrolidone good supplier in Chi
3355-31-5
1400634-44-7
6020-87-7
134-62-3
110-26-9
2381089-83-2
137-08-6
56-84-8
68333-79-9
13463-67-7
51115-67-4
142217-69-4
18472-51-0
27176-87-0
86532-26-5
458-37-7
210155-39-8
144-62-7
22888-70-6
122-99-6
540737-29-9
272778-12-8
55289-06-0
497-30-3

Article Doi