Archiv der Pharmazie p. 247 - 255 (1995)
Update date:2022-09-26
Topics:
Gorlitzer
Wilpert
Rubsamen-Waigmann
Suhartono
Wang
Immelmann
Starting from the commercially available 6-methyl-2-pyridylamine (1) the pyrido[3,2-e][1,4]diazepine 14a was synthesized in 12 steps with 7% total yield. 14a, the N-methyl derivative 14b, the thiolactam 15a, the amidine 16, and the 1,2,4-triazole 17 were tested for anti-HIV-1-activity. None of the compounds tested possesses antiviral activity comparable to that of zidovudine (3'-azido-3'-desoxythymidine = AZT).
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Doi:10.1016/0040-4039(95)00819-X
(1995)Doi:10.1016/0022-328X(95)05215-B
(1995)Doi:10.1021/jo400954p
(2013)Doi:10.1039/DT9950000931
(1995)Doi:10.1021/jo026853m
(2003)Doi:10.1021/om9602771
(1996)
