Enantio- and diastereocontrolled synthesis of epibatidine analogues

DOI: 10.1248/cpb.43.901

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 901 - 903 (1995)

Update date:2022-07-30

Topics:

Authors:

Hiroya Hiroya

Uwai Uwai

Ogasawara

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.43.901

Three structural analogues of a potent non-opiate analgesic alkaloid epibatidine have been synthesized in optically pure forms in enantio- and diastereo-controlled ways using a chiral 2,5-cyclohexadiene-1,4-diol synthon.

Full text of DOI:10.1248/cpb.43.901

NII-Electronic Library Service

Products guided by the article

Product name:(1S,4R,4aS,7S,8R,8aR)-8-Methoxymethoxy-7-(3-methoxy-phenyl)-4,4a,6,7,8,8a-hexahydro-1H-1,4-methano-naphthalen-5-one

Cas No:167387-10-2

R&D Labs maybe for 167387-10-2

Tianjin Emulsion Science&Technology Development Co.,Ltd

Contact:13901380442

Address:Vake Garden New Town New Yi Bai Road Beichen District Tianjin,China
jiangsu senxuan pharmaceutical and chemical co.,ltd

Contact:86-523-87982810

Address:hongqiao industrial zone,taixing,jiangsu china
Suzhou Chenke Biotech Co., Ltd.

Contact:+86-18662408853

Address:NO.150, Renai Road, Suzhou Industrial Park
Feis International Trade Co,. Ltd

Contact:13961823444-18235944442

Address:Wuxi jiangsu
Zhushan County Tianxin Pharmaceutical & Chemical Co., Ltd.

Contact:0086-719-4224892

Address:Tutang Road, Chengguan Town, Zhushan County, Hubei Province

Relevant to this article

Ruthenium(II) 8-quinolinolates: Synthesis, characterization, crystal structure and catalysis in the synthesis of 2-oxazolines

Doi:10.1016/j.jorganchem.2015.06.005
(2015)
Formation of thiazyl radicals by the thermolysis and photolysis of sulfur-nitrogen bicycles RCN₅S₃

Doi:10.1016/j.mencom.2007.06.005
(2007)
Doi:10.1021/jo01254a010
(1969)
Doi:10.1021/jo01068a041
(1961)
Organocatalytic Enantioselective Conia-Ene-Type Carbocyclization of Ynamide Cyclohexanones: Regiodivergent Synthesis of Morphans and Normorphans

Doi:10.1002/anie.201908495
(2019)
Chemoselective (trans)thioacetalization of carbonyl compounds with a reusable lewis acid-surfactant-combined copper bis(dodecyl sulfate) catalyst in water

Doi:10.1055/s-0029-1218693
(2010)

Article Doi