Enantio- and diastereocontrolled synthesis of epibatidine analogues

DOI: 10.1248/cpb.43.901

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 901 - 903 (1995)

Update date:2022-07-30

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Authors:

Hiroya Hiroya

Uwai Uwai

Ogasawara

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Article abstract of DOI:10.1248/cpb.43.901

Three structural analogues of a potent non-opiate analgesic alkaloid epibatidine have been synthesized in optically pure forms in enantio- and diastereo-controlled ways using a chiral 2,5-cyclohexadiene-1,4-diol synthon.

Full text of DOI:10.1248/cpb.43.901

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