Synthesis and biological activity of heterocyclic aminophosphonates

Article abstract of DOI:10.1080/10426509908546274

A variety of synthetic methods for preparation of heterocyclic aminophosphonates is presented; which are concerning furyl, thienyl, pyrryl and pyridyl derivatives of aminomethanephosphonic acid and also phosphonic analogues of proline and homoproline. The obtained heterocyclic aminophosphonates were used as starting materials for synthesis of some peptidyl phosphonates. The compounds were evaluated as inhibitors of serine proteases. Most of the obtained heterocyclic aminophosphonates were preliminary tested as potential herbicides against selected plants, and some of them showed the herbicidal activity.

Full text of DOI:10.1080/10426509908546274

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Phosphorus, Sulfur, and
Silicon and the Related
Elements
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Synthesis and Biological
Activity of Heterocyclic
Aminophosphonates
Bogdan Boduszek
a Institute of Organic Chemistry,
Biochemistry and Biotechnology,
Wroclaw University of Technology, 50–370
Wroclaw, Poland
Version of record first published: 17 Mar
2008
To cite this article: Bogdan Boduszek (1999): Synthesis and Biological
Activity of Heterocyclic Aminophosphonates, Phosphorus, Sulfur, and
Silicon and the Related Elements, 144:1, 433-436
To link to this article: http://dx.doi.org/10.1080/10426509908546274
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