
Bioorganic and Medicinal Chemistry Letters p. 161 - 164 (1996)
Update date:2022-07-30
Topics:
Chan, Chuen
Cocker, J. Derek
Davies, H. Geoffrey
Gore, Andrea
Green, Richard H.
Two novel indolizidine analogues, (7a) and (7b), of the substance P antagonist CP 99,994 have been prepared. Possible conformational factors for their low biological activity are discussed.
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