Synthesis of a model bicyclic C-O-D-O-E ring of vancomycin by a one-pot, double SNAr based macrocyclization

DOI: 10.1039/cc9960001029

Source and publish data:

Chemical Communications p. 1029 - 1030 (1996)

Update date:2022-07-30

Topics:

Authors:

Beugelmans, Rene

Bois-Choussy, Michele

Vergne, Caroline

Bouillon, Jean-Philippe

Zhu, Jieping

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1039/cc9960001029

Double cyclization of linear pentapeptide 3 by treatment with CsF in DMF at -5°C gives a model bicyclic CODOE ring 2 of vancomycin in a one-pot fashion.

Full text of DOI:10.1039/cc9960001029

View Article Online / Journal Homepage / Table of Contents for this issue

View Article Online

Products guided by the article

Product name:(S)-2-[(R)-2-tert-Butoxycarbonylamino-3-(4-fluoro-3-nitro-phenyl)-propionylamino]-propionic acid

Cas No:178744-44-0

R&D Labs maybe for 178744-44-0

Acros Pharmatech Limited

website:http://www.acrospharmatech.com

Contact:+1-3234804688

Address:Flat/RM 1502,Easey Commercial building 253-261 Hennessy Road,Wanchai，HongKong
Pengchen New Material Technology Co., Ltd.

Contact:+86-512-63680537

Address:99.6 km of national road 318, Meiyan Community,Pingwang Town, Wujiang District, Suzhou 215225
Hangzhou Neway Chemicals Co., Ltd.

Contact:+86-571-85095566

Address:Room 803, Qinglian Bldg, No 139 Qingchun Road, Hangzhou, Zhejiang China
Chinapeptides Co,. Ltd

Contact:+86-021-50792271

Address:Building 24A, 300 Chuantu Road, Chuansha, Pudong new area, Shanghai, China, 201202
Changzhou LanXu Chemical Co.,ltd.(expird)

Contact:86-0519-86330911,13656129734,15261186386

Address:Room 524, Depart.Chemical, Changzhou Science and Eductaion town, Jiangsu, China;Factory: Haian Fine Chemical Industry Park,Nantong,Jiangsu,China

Relevant to this article

Palladium-catalyzed annulation of alkynes with ortho -halide-containing benzyl alcohols in aqueous medium

Doi:10.1021/jo501444g
(2014)
Doi:10.1007/BF00481588
()
Quantitative description of structural effects on the stability of gold(I) carbenes

Doi:10.1002/chem.201403988
(2014)
Highly Deformed o-Carborane Functionalised Non-linear Polycyclic Aromatics with Exceptionally Long C?C Bonds

Doi:10.1002/chem.202004517
(2021)
Tandem Beckmann and Huisgen-White rearrangement as an alternative to the Baeyer-Villiger oxidation of the bicyclo[3.3.1]nonane system: First asymmetric synthesis of (-)-dihydropalustramic acid. X-Ray molecular structure of 2β-ethyl-9-phenylsulfonyl-9-azabicyclo[3.3.1]nonan-3-one

Doi:10.1039/P19960001567
(1996)
Synthesis of Diaryliodonium Salts Having Pentafluorosulfanylarenes and Their Application to Electrophilic Pentafluorosulfanylarylation of C-, O-, N-, and S-Nucleophiles

Doi:10.1021/acs.orglett.5b01323
(2015)

Article Doi