A new indole synthesis via [3 + 3] annulation of 2-(benzotriazol-1-ylmethyl)pyrroles with α,β-unsaturated aldehydes and ketones

DOI: 10.1016/0040-4039(96)01216-6

Source and publish data:

Tetrahedron Letters p. 5641 - 5644 (1996)

Update date:2022-08-05

Topics:

Authors:

Katritzky, Alan R.

Levell, Julian R.

Li, Jianqing

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0040-4039(96)01216-6

Poly-substituted indoles are readily accessible from substituted 2-(benzotriazol-1-ylmethyl)pyrroles by lithiation, reaction with α,β-unsaturated aldehydes and ketones, and subsequent facile dehydrobenzotriazolylation-cyclodehydration. The substituted 2-(

Full text of DOI:10.1016/0040-4039(96)01216-6

Products guided by the article

Product name:1-(1-tert-Butyl-4-phenyl-1H-pyrrol-2-ylmethyl)-1H-benzotriazole

Cas No:180271-48-1

R&D Labs maybe for 180271-48-1

Liao Cheng All Win Chemicals Co.,LTD

Contact:86+0635-2991582

Address:Room 402,Unit 1,No.27 building.Zhong tong shi dai haoyuan,liaocheng city,Shan dong Province.China
Chengdu ZY Biochemical Technology Co., LTD

Contact:0086-28-88680086

Address:170 Qingpu Road, Shouan Town, Pujiang County
Xi'an yuanfar international trade company

website:https://www.yuanfarchemical.com

Contact:86-029-88745613 ext 828

Address:Floor19th ,B Building, Oak Block,No.36 South Fenghui Road, Dev. Zone of High-Tech Ind.,Xi’an, China
Yancheng Creator Chemical Co., Ltd

Contact:0086-515-88710008 88710068 88710858 88710868

Address:No.21 Renming Road, Longgang Town, Yandu County,Yancheng City
SHANDONG CREDAGRI CHEMICAL CO., LTD.

Contact:+86-531-88872050

Address:ROOM 601A, BUILDING 2, SHUNTAI SQUARE, NO. 2000 SHUNHUA ROAD, HI-TECH DEVELOPMENT ZONE, JINAN, CHINA.

Relevant to this article

Capacity of thiourea Schiff base esters as multifunctional additives: synthesis, characterization and performance evaluation in polyol

Doi:10.1039/c5ra13507a
(2015)
Doi:10.1007/BF00843948
()
Synthesis, Protonation and Co-ordination Abilities of the Open-chain Polyamine 4,8,11,15-Tetraazaoctadecane-1,18-diamine

Doi:10.1039/DT9940000637
(1994)
Cis-trans isomerization of a cyclopropyl radical trap catalyzed by extradiol catechol dioxygenases: Evidence for a semiquinone intermediate

Doi:10.1021/ja9607704
(1996)
Synthesis of new 1H-tetrazoles and 1,2,3-triazoles via reactions of 3(,5)-di(chloro-2H-1,4-(benz)oxazin-2-ones with sodium azide or diazocompounds

Doi:10.1016/0040-4020(96)00423-1
(1996)
A practical and efficient route for synthesis of 6-aminomethyl-4-oxo- 4,5,6,7-tetrahydroindoles as new CNS agent precursors

Doi:10.1016/0040-4039(96)01028-3
(1996)

Article Doi