A practical and efficient route for synthesis of 6-aminomethyl-4-oxo- 4,5,6,7-tetrahydroindoles as new CNS agent precursors

DOI: 10.1016/0040-4039(96)01028-3

Source and publish data:

Tetrahedron Letters p. 5171 - 5174 (1996)

Update date:2022-08-05

Topics:

Authors:

Masaguer, Christian F.

Ravina, Enrique

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Article abstract of DOI:10.1016/0040-4039(96)01028-3

Starting from 2,5-dimethoxybenzoic acid we described a practical and efficient route for synthesis of 6-aminomethyl-4-oxotetrahydroindoles with good to acceptable overall yields of 50-30%.

Full text of DOI:10.1016/0040-4039(96)01028-3

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