A practical and efficient route for synthesis of 6-aminomethyl-4-oxo- 4,5,6,7-tetrahydroindoles as new CNS agent precursors

DOI: 10.1016/0040-4039(96)01028-3

Source and publish data:

Tetrahedron Letters p. 5171 - 5174 (1996)

Update date:2022-08-05

Topics:

Authors:

Masaguer, Christian F.

Ravina, Enrique

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0040-4039(96)01028-3

Starting from 2,5-dimethoxybenzoic acid we described a practical and efficient route for synthesis of 6-aminomethyl-4-oxotetrahydroindoles with good to acceptable overall yields of 50-30%.

Full text of DOI:10.1016/0040-4039(96)01028-3

Products guided by the article

Product name:1-(3,5-Dimethoxy-cyclohexa-2,5-dienylmethyl)-piperazine

Cas No:181047-38-1

R&D Labs maybe for 181047-38-1

Advanced Biotech

Contact:+1-973-357-0577

Address:10 Taft Rd.
Changzhou Litong Chemical Co., Ltd.

website:http://www.litonchem.com/

Contact:+86-519-86301238

Address:Laoba Rd, Hutang town Changzhou Jiangsu
MINS GROUP CO.,LIMITED

Contact:18669908765

Address:Zibo City, Shandong Province, P.R.China
Aecochem Corp.

website:http://www.aecochemical.com

Contact:+86-592 599 8717

Address:No 611 Sishui Road,Huli
Changzhou Sunlight Pharmaceutical Co., Ltd.

Contact:+86-519-83131668;83139028;83138042;83137041

Address:JiuliStreet, Benniu Town Changzhou City, Jiangsu Province

Relevant to this article

Stereoconservative synthesis of orthogonally protected γ-functionalized amino acids using N-tritylserine derivatives

Doi:10.1021/jo960624g
(1996)
Total synthesis of (±)-deethylibophyllidine: Studies of a Fischer indolization route and a successful approach via a Pummerer rearrangement/thionium ion-mediated indole cyclization

Doi:10.1021/jo960848z
(1996)
Doi:10.1039/j39660000566
(1966)
Conversion of η²-phosphinocarbene complexes into tungstaphosphabicyclo[1.1.0]butanone units

Doi:10.1016/S0022-328X(97)00632-3
(1998)
A Dihydrogen Complex, 2-H2)(CO)(quS)(PPh3)2>+, in Equilibrium with its Coordinated Thiol Tautomer (quS = quinoline-8-thiolate)

Doi:10.1039/c39950000625
(1995)
Chemistry of H2O⁺ with C2F4, C2F6, and CF3X (X = F, Cl, Br, I)

Doi:10.1021/j100186a050
(1992)

Article Doi