An efficient synthesis of magallanesine using [1,2]-Meisenheimer rearrangement and Heck cyclization

Article abstract of DOI:10.1016/0040-4020(96)00900-3

A straightforward total synthesis of magallanesine 1 was accomplished from readily available isoquinolineacetate 14. This synthesis is emphasized by the following two points; i. the [1,2]-Meisenheimer rearrangement of the azetidine N-oxide 22 for the prep