Bioorganic and Medicinal Chemistry Letters p. 213 - 218 (1997)
Update date:2022-08-03
Topics: Synthesis Ligand Optimization binding affinity Functional Characterization Experimental Nonpeptidic agonist
De Laszlo
Allen
Li
Ondeyka
Rivero
Malkowitz
Molineaux
Siciliano
Springer
Greenlee
Mantlo
The structural optimization for binding affinity and attempted modification of agonist function of a nonpeptide ligand of the human C5a receptor is described.
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Doi:10.1016/S0022-328X(97)00441-5
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(1997)Doi:10.1016/S0960-894X(99)00196-1
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(2018)Doi:10.1055/s-0029-1216973
(2009)Doi:10.1039/a606551a
(1997)