Tetrahedron Letters p. 1161 - 1164 (1997)
Update date:2022-08-03
Topics:
Gray, Nathanael S.
Kwon, Soojin
Schultz, Peter G.
A method for the combinatorial synthesis of 2,9-substituted purines using a Mitsunobu reaction to alkylate the N-9 position and an amination reaction to install amines at the C-2 position has been developed.
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