Azapeptides as inhibitors and active site titrants for cysteine proteinases

Article abstract of DOI:10.1021/jm970802d

Ester and amide derivatives of α-azaglycine (carbazic acid, H₂NHCOOH), α-azaalanine, and α-azaphenylalanine (i.e., AC-L-Phe-NHN(R)CO-X, where X = H, CH₃, or CH₂Ph, respectively) were synthesized and evaluated as inhibitors