New efficient syntheses of α-difluoromethyl- and α-trifluoromethyl-ornithine

DOI: 10.1016/S0040-4039(97)01344-0

Source and publish data:

Tetrahedron Letters p. 5965 - 5966 (1997)

Update date:2022-08-03

Topics:

Authors:

Osipov, Sergey N.

Golubev, Alexander S.

Sewald, Norbert

Burger, Klaus

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(97)01344-0

A new efficient method for the preparation of ornithine derivatives 3-5 is described. The key step of the synthesis is the regioselective alkylation of imine 2 with propargyl amine 1.

Full text of DOI:10.1016/S0040-4039(97)01344-0

Products guided by the article

Product name:3-Pentynoic acid, 5-amino-2-(difluoromethyl)-2-[[(phenylmethoxy)carbonyl]amino]-, methyl ester

Cas No:195195-99-4

R&D Labs maybe for 195195-99-4

Yuan Shi(SuQian)Biotechnology Co.,Ltd

website:http://www.yuanshibio.com

Contact:+86-527-84226672

Address:jiangsu suqian
Jinzhou Jiutai Pharmaceutical Co.,Ltd

Contact:+86-0416-5179890

Address:No.41, Taianli, Taihe District, Jinzhou, Liaoning
Dalian Synco Chemical Co., Ltd.

Contact:+86-411-83635150

Address:Rm 1004, 24, Tangshan Street, Dalian
Jiaxing Trustworthy Import And Export Co.,Ltd

Contact:+86-573-82030555

Address:Room 1202, Unit B, Charming plaza,No.1558 East Zhongshan Road , Jiaxing City, Zhejiang Province, China.
Wuhan Sunrise Pharmaceutical Technology Co., Ltd

Contact:+86-27-83314682

Address:Room 340, New material Industrial base No.17, Gu Tian Five Lu , Qiaokou District, Wuhan , China

Relevant to this article

Polyethers with phosphate pendant groups by monomer activated anionic ring opening polymerization: Syntheses, characterization and their lithium-ion conductivities

Doi:10.1016/j.polymer.2013.12.005
(2014)
Reaction of alkynes with Rh₄(CO)₁₂. A mid-infrared vibrational and kinetic study of (μ₄-η²-alkyne) Rh₄(CO)₈(μ-CO)₂

Doi:10.1021/om0510019
(2006)
Vibrational and thermodynamic properties and molecular motions in the incommensurate crystal of morpholinium tetrafluoroborate studied by ¹H NMR

Doi:10.1016/j.chemphys.2011.01.002
(2011)
Efficient asymmetric synthesis of phosphatidyl-D-myo-inositol 3,4,5- trisphosphate

Doi:10.1248/cpb.45.1521
(1997)
Synthesis, biological evaluation and molecular docking study of 2-substituted-4, 6-diarylpyrimidines as α-glucosidase inhibitors

Doi:10.3390/molecules22111865
(2017)
Azamorphinan and related compounds. I. A synthesis of 2-hydroxy-N-methyl-9-azamorphinan (studies on the syntheses of heterocyclic compounds. CCXIV.

Doi:10.1248/cpb.16.296
(1968)

Article Doi