Investigation on some reactions of saccharinyl benzoic acid azides

Article abstract of DOI:10.1080/10426509708040505

Saccharinyl benzole acid azides 2a-c were used to synthesize a number of noncondensed heterocyclic systems. Thus azides 2a or 2c reacted with glycine to give 1,3-oxazolin-5-one derivatives 3a and 3b. However azide 2b reacted to give diaryl urea derivative which was easily cyclized to give imidazol -2,5- dione (6). Also azides 2a-c reacted with glycolic acid to give 1,3-oxazolin -2,5-dione derivatives (7a-c) and with aroyl hydrazines to give the corresponding hydrazides (8a-f) which were cyclized to 1,3,5-oxadiazole derivatives (9a-f).

Full text of DOI:10.1080/10426509708040505

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Phosphorus, Sulfur, and Silicon and the
Related Elements
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INVESTIGATION ON SOME REACTIONS OF
SACCHARINYL BENZOIC ACID AZIDES
M. M. H. Arief a
a Chemistry Department, Faculty of Sciencec , Benha University , Benha,
Egypt
Published online: 04 Oct 2006.
To cite this article: M. M. H. Arief (1997) INVESTIGATION ON SOME REACTIONS OF SACCHARINYL
BENZOIC ACID AZIDES, Phosphorus, Sulfur, and Silicon and the Related Elements, 127:1, 159-165, DOI:
10.1080/10426509708040505
To link to this article: http://dx.doi.org/10.1080/10426509708040505
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