
Journal of Medicinal Chemistry p. 2218 - 2226 (1999)
Update date:2022-08-04
Topics:
Costanzo, Annarella
Guerrini, Gabriella
Ciciani, Giovanna
Bruni, Fabrizio
Selleri, Silvia
Costa, Barbara
Martini, Claudia
Lucacchini, Antonio
Malmberg Aiello, Petra
Ipponi, Alessandra
The synthesis of new 3-heteroaryl-8-chloropyrazolo[5,1- c][1,2,4]benzotriazine 5-oxides and their binding activities at the central benzodiazepine receptor (BZR) are reported. The derivatives substituted at the 3-position with electron-rich five-membered
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(1999)