First fatty acylated dipeptides to affect muscarinic receptor ligand binding

Article abstract of DOI:10.1016/S0960-894X(99)00604-6

Fatty acylated dipeptides homologous to G(i)α N-termini affect ligand binding to muscarinic acetylcholine receptors. Myristylglycine-serine containing dipeptides decrease antagonist binding at both M₁ and Ms muscarinic receptors. Palmitate on t