A new class of conformationally rigid analogues of 4-amino-5- halopentanoic acids, potent inactivators of γ-aminobutyric acid aminotransferase

DOI: 10.1021/jm9904755

Source and publish data:

Journal of Medicinal Chemistry p. 706 - 720 (2000)

Update date:2022-08-05

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Authors:

Qiu, Jian

Silverman, Richard B.

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Article abstract of DOI:10.1021/jm9904755

Recently, we found (Qiu, J.; Pingsterhaus, J. M.; Silverman, R. B. J. Med. Chem. 1999, 42, 4725-4728) that conformationally rigid analogues of the GABA aminotransferase (GABA-AT) inactivator vigabatrin were not inactivators of GABA-AT. To determine if thi

Full text of DOI:10.1021/jm9904755

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