Bioorganic and Medicinal Chemistry Letters p. 1767 - 1770 (2003)
Update date:2022-08-04
Topics:
Chai, Wenying
Breitenbucher, J. Guy
Kwok, Annette
Li, Xiaobing
Wong, Victoria
Carruthers, Nicholas I.
Lovenberg, Timothy W.
Mazur, Curt
Wilson, Sandy J.
Axe, Frank U.
Jones, Todd K.
Continued exploration of the SAR around the lead imidazopyridine histamine H3 antagonist 1 has led to the discovery of several related series of heterocyclic histamine H3 antagonists. The synthesis and SAR of indolizine, indole and p
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