Journal of labelled compounds and radiopharmaceuticals p. 627 - 634 (1994)
Update date:2022-08-03
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Ekhato
Huang
Carbon-14 labeled 3,5-dihydro-5-methyl-1(2H)-isoquinolinone, a potent inhibitor of poly(ADP-ribose) polymerase (ADPRP) was prepared from 1-bromo-2-methylbenzene in 7.8 % overall yield. The C-14 label was introduced from Ba(l)4CO3 via
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